(Q35016160)

5 August 2017

title

Why are membrane targets discovered by phenotypic screens and genome sequencing in Mycobacterium tuberculosis? (English)

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Mycobacterium tuberculosis

5 August 2017

main subject

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author name string

Robert C Goldman

series ordinal

1

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5 August 2017

publication date

18 September 2013

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5 August 2017

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5 August 2017

volume

93

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5 August 2017

issue

6

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5 August 2017

page(s)

569-588

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Totally drug-resistant tuberculosis in India.

5 August 2017

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7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Property distributions: differences between drugs, natural products, and molecules from combinatorial chemistry

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Scaffold architecture and pharmacophoric properties of natural products and trade drugs: application in the design of natural product-based combinatorial libraries

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Chemoinformatic analysis of combinatorial libraries, drugs, natural products, and molecular libraries small molecule repository

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

A structure-permeability study of small drug-like molecules.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

A practical view of 'druggability'.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Selection criteria for drug-like compounds

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Molecular properties that influence the oral bioavailability of drug candidates

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

A comparison of physiochemical property profiles of development and marketed oral drugs

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Going further than Lipinski's rule in drug design

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Ligand Efficiency Indices (LEIs): More than a Simple Efficiency Yardstick

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Ligand efficiency indices for an effective mapping of chemico-biological space: the concept of an atlas-like representation.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

AtlasCBS: a web server to map and explore chemico-biological space.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

A sorcerer's apprentice and The Rule of Five: from rule-of-thumb to commandment and beyond

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Strong Inference: Certain systematic methods of scientific thinking may produce much more rapid progress than others

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Ask the experts: past, present and future of the rule of five

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Chris Lipinski discusses life and chemistry after the Rule of Five.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Let's get specific: the relationship between specificity and affinity

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Chlorobiphenyl-desleucyl-vancomycin inhibits the transglycosylation process required for peptidoglycan synthesis in bacteria in the absence of dipeptide binding

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Synthesis of hydrophobic N'-mono and N',N"-double alkylated eremomycins inhibiting the transglycosylation stage of bacterial cell wall biosynthesis.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Synthesis and mode of action of hydrophobic derivatives of the glycopeptide antibiotic eremomycin and des-(N-methyl-D-leucyl)eremomycin against glycopeptide-sensitive and -resistant bacteria

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Genetic basis for activity differences between vancomycin and glycolipid derivatives of vancomycin.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Ligand binding in the conserved interhelical loop of CorA, a magnesium transporter from Mycobacterium tuberculosis

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Construction of a series of vectors for high throughput cloning and expression screening of membrane proteins from Mycobacterium tuberculosis

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

1H, 15N and 13C backbone resonance assignment of Rv1567c, an integral membrane protein from Mycobacterium tuberculosis

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Uniformly aligned full-length membrane proteins in liquid crystalline bilayers for structural characterization

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Expression of membrane proteins from Mycobacterium tuberculosis in Escherichia coli as fusions with maltose binding protein

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Structural biology of transmembrane domains: efficient production and characterization of transmembrane peptides by NMR.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Identification of Mycobacterium tuberculosis H37Rv integral membrane proteins by one-dimensional gel electrophoresis and liquid chromatography electrospray ionization tandem mass spectrometry

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Cloning and expression of multiple integral membrane proteins from Mycobacterium tuberculosis in Escherichia coli

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Daptomycin: a review of properties, clinical use, drug delivery and resistance

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Telavancin: a novel lipoglycopeptide

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Amphotericin B membrane action: role for two types of ion channels in eliciting cell survival and lethal effects

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Cellular pharmacokinetics of telavancin, a novel lipoglycopeptide antibiotic, and analysis of lysosomal changes in cultured eukaryotic cells (J774 mouse macrophages and rat embryonic fibroblasts).

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Mixed-lipid storage disorder induced in macrophages and fibroblasts by oritavancin (LY333328), a new glycopeptide antibiotic with exceptional cellular accumulation

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Identification of a small molecule with activity against drug-resistant and persistent tuberculosis

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

Accumulation of norfloxacin by Mycobacterium aurum and Mycobacterium smegmatis

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

inferred from DOI database lookup

7 January 2021

based on heuristic

Porins in the cell wall of Mycobacterium tuberculosis.

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

inferred from DOI database lookup

7 January 2021

based on heuristic

Mefloquine is active in vitro and in vivo against Mycobacterium avium complex

1 reference

https://api.crossref.org/works/10.1016%2FJ.TUBE.2013.09.003

inferred from DOI database lookup

7 January 2021

based on heuristic

Identifiers

DOI

10.1016/J.TUBE.2013.09.003

1 reference

5 August 2017

1 reference