(Q36242609)

English

Mutagenesis and computer modeling studies of a GPCR conserved residue W5.43(194) in ligand recognition and signal transduction for CB2 receptor

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

Mutagenesis and computer modeling studies of a GPCR conserved residue W5.43(194) in ligand recognition and signal transduction for CB2 receptor (English)

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

G protein-coupled receptor

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5

object named as

John S Lazo

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

author name string

Yuxun Zhang

1

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

Zhaojun Xie

2

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

Lirong Wang

3

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

Brielle Schreiter

4

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

Jurg Gertsch

6

1 reference

Europe PubMed Central

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13 August 2017

Xiang-Qun Xie

7

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Europe PubMed Central

PMC publication ID

13 August 2017

publication date

1 May 2011

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

International Immunopharmacology

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Europe PubMed Central

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13 August 2017

11

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Europe PubMed Central

PMC publication ID

13 August 2017

9

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

1303-1310

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

Identification of compounds that potentiate CREB signaling as possible enhancers of long-term memory

1 reference

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1 October 2017

Residues accessible in the binding-site crevice of transmembrane helix 6 of the CB2 cannabinoid receptor

1 reference

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1 October 2017

Ligand-binding architecture of human CB2 cannabinoid receptor: evidence for receptor subtype-specific binding motif and modeling GPCR activation.

1 reference

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Beta-caryophyllene is a dietary cannabinoid

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The preference of tryptophan for membrane interfaces: insights from N-methylation of tryptophans in gramicidin channels

1 reference

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Cannabinoid CB1 and CB2 receptor ligand specificity and the development of CB2-selective agonists.

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Targeting the cannabinoid CB2 receptor: modelling and structural determinants of CB2 selective ligands

1 reference

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CB2 receptors as new therapeutic targets for liver diseases

1 reference

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GPCR structure-based virtual screening approach for CB2 antagonist search

1 reference

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The effects of charge-neutralizing mutation D6.30N on the functions of CB1 and CB2 cannabinoid receptors

1 reference

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A cannabinoid receptor 1 mutation proximal to the DRY motif results in constitutive activity and reveals intramolecular interactions involved in receptor activation

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Cannabinoid receptors and their ligands: ligand-ligand and ligand-receptor modeling approaches

1 reference

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Alkylamides from Echinacea are a new class of cannabinomimetics. Cannabinoid type 2 receptor-dependent and -independent immunomodulatory effects

1 reference

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1 October 2017

Cannabinoid CB2/CB1 selectivity. Receptor modeling and automated docking analysis

1 reference

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1 October 2017

Targeting the cannabinoid CB2 receptor: mutations, modeling and development of CB2 selective ligands.

1 reference

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1 October 2017

Cysteine 2.59(89) in the second transmembrane domain of human CB2 receptor is accessible within the ligand binding crevice: evidence for possible CB2 deviation from a rhodopsin template.

1 reference

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1 October 2017

Structural mimicry in class A G protein-coupled receptor rotamer toggle switches: the importance of the F3.36(201)/W6.48(357) interaction in cannabinoid CB1 receptor activation

1 reference

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1 October 2017

Anandamide initiates Ca(2+) signaling via CB2 receptor linked to phospholipase C in calf pulmonary endothelial cells

1 reference

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1 October 2017

3D structural model of the G‐protein‐coupled cannabinoid CB2 receptor

1 reference

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1 October 2017

Mutational analysis and molecular modelling of the antagonist SR 144528 binding site on the human cannabinoid CB(2) receptor

1 reference

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1 October 2017

Role of a conserved lysine residue in the peripheral cannabinoid receptor (CB2): evidence for subtype specificity

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3445262

1 October 2017

SR 144528, an antagonist for the peripheral cannabinoid receptor that behaves as an inverse agonist.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3445262

1 October 2017

Signaling pathway associated with stimulation of CB2 peripheral cannabinoid receptor. Involvement of both mitogen-activated protein kinase and induction of Krox-24 expression

1 reference

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1 October 2017

A mutation-induced activated state of the beta 2-adrenergic receptor. Extending the ternary complex model

1 reference

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1 October 2017

Expression of central and peripheral cannabinoid receptors in human immune tissues and leukocyte subpopulations

1 reference

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1 October 2017

Concurrent stimulation of cannabinoid CB1 and dopamine D2 receptors augments cAMP accumulation in striatal neurons: evidence for a Gs linkage to the CB1 receptor.

1 reference

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Surflex-Dock 2.1: robust performance from ligand energetic modeling, ring flexibility, and knowledge-based search

1 reference

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Novel 4-oxo-1,4-dihydroquinoline-3-carboxamide derivatives as new CB2 cannabinoid receptors agonists: synthesis, pharmacological properties and molecular modeling.

1 reference

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Virtual screening of novel CB2 ligands using a comparative model of the human cannabinoid CB2 receptor.

1 reference

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A novel cannabinoid peripheral cannabinoid receptor-selective inverse agonist blocks leukocyte recruitment in vivo

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Chemical modification of the naphthoyl 3-position of JWH-015: in search of a fluorescent probe to the cannabinoid CB2 receptor.

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22 September 2018

Cannabinoid receptor activation differentially regulates the various adenylyl cyclase isozymes

1 reference

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Gi protein modulation induced by a selective inverse agonist for the peripheral cannabinoid receptor CB2: implication for intracellular signalization cross-regulation

1 reference

https://pubmed.ncbi.nlm.nih.gov/21539938

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The difference between the CB(1) and CB(2) cannabinoid receptors at position 5.46 is crucial for the selectivity of WIN55212-2 for CB(2)

1 reference

https://pubmed.ncbi.nlm.nih.gov/21539938

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Homology models of the cannabinoid CB1 and CB2 receptors. A docking analysis study

1 reference

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1016/J.INTIMP.2011.04.013

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

ResearchGate publication ID

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