(Q37765564)

22 August 2017

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title

Recent advances in the development of novel glucocorticoid receptor modulators (English)

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22 August 2017

Michael Berlin

1

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22 August 2017

language of work or name

English

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publication date

1 July 2010

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Expert Opinion on Therapeutic Patents

22 August 2017

published in

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22 August 2017

volume

20

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22 August 2017

issue

7

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22 August 2017

page(s)

855-873

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Effects of glucocorticoids on inflammation and arthritis.

22 August 2017

cites work

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Glucocorticoid-induced apoptosis and glucocorticoid resistance: molecular mechanisms and clinical relevance.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Mechanisms involved in the side effects of glucocorticoids

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Glucocorticoid dysregulations and their clinical correlates. From receptors to therapeutics

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Glucocorticoid action and the development of selective glucocorticoid receptor ligands

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Non-steroidal glucocorticoid receptor antagonists: the race to replace RU-486 for anti-glucocorticoid therapy

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Recent developments in the discovery of selective glucocorticoid receptor modulators (SGRMs).

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Recent progress in the discovery of novel glucocorticoid receptor modulators

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Genomic and nongenomic effects of glucocorticoids

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Novel insights into mechanisms of glucocorticoid action and the development of new glucocorticoid receptor ligands

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Modelling the glucocorticoid receptor and producing therapeutic agents with anti-inflammatory effects but reduced side-effects

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Glucocorticoids, metabolism and metabolic diseases.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Controlling nuclear receptors: the circular logic of cofactor cycles

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Ligand-selective transactivation and transrepression via the glucocorticoid receptor: role of cofactor interaction

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Modulation of glucocorticoid receptor induction properties by cofactors in peripheral blood mononuclear cells

21 January 2018

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Selective glucocorticoid receptor agonists (SEGRAs): novel ligands with an improved therapeutic index.

21 January 2018

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DNA binding of the glucocorticoid receptor is not essential for survival

21 January 2018

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Repression of inflammatory responses in the absence of DNA binding by the glucocorticoid receptor

21 January 2018

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Dissociation of transactivation from transrepression by a selective glucocorticoid receptor agonist leads to separation of therapeutic effects from side effects

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Principles for modulation of the nuclear receptor superfamily

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

A single amino acid change in the first zinc finger of the DNA binding domain of the glucocorticoid receptor regulates differential promoter selectivity.

21 January 2018

1 reference

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New perspectives in the treatment of Cushing's syndrome

21 January 2018

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Modulation of glucocorticoid action and the treatment of type-2 diabetes

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Characterization of a novel non-steroidal glucocorticoid receptor antagonist

21 January 2018

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Liver-selective glucocorticoid receptor antagonism decreases glucose production and increases glucose disposal, ameliorating insulin resistance

21 January 2018

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New and established topical corticosteroids in dermatology: clinical pharmacology and therapeutic use.

21 January 2018

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Corticosteroid design for the treatment of asthma: structural insights and the therapeutic potential of soft corticosteroids

21 January 2018

1 reference

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Characterization of ZK 245186, a novel, selective glucocorticoid receptor agonist for the topical treatment of inflammatory skin diseases

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Doubling the Size of the Glucocorticoid Receptor Ligand Binding Pocket by Deacylcortivazol

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

The first X-ray crystal structure of the glucocorticoid receptor bound to a non-steroidal agonist

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Discovery of novel dihydro-9,10-ethano-anthracene carboxamides as glucocorticoid receptor modulators

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

Discovery of potent, nonsteroidal, and highly selective glucocorticoid receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.493876

A role for proteinase-activated receptor-1 in inflammatory bowel diseases

21 January 2018

1 reference

30 December 2023

https://opencitations.net/index/api/v1/citations/10.1172/JCI21689

Identifiers

DOI

10.1517/13543776.2010.493876

1 reference

22 August 2017

1 reference