(Q40052763)

English

Point mutations in the second extracellular loop of the histamine H2 receptor do not affect the species-selective activity of guanidine-type agonists

scientific article published on 13 November 2007

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

Point mutations in the second extracellular loop of the histamine H2 receptor do not affect the species-selective activity of guanidine-type agonists (English)

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

author name string

Hendrik Preuss

1

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

Prasanta Ghorai

2

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

Anja Kraus

3

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

Stefan Dove

4

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

Armin Buschauer

5

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

Roland Seifert

6

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

publication date

13 November 2007

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

Naunyn-Schmiedeberg's Archives of Pharmacology

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

376

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

4

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

253-264

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

https://scigraph.springernature.com/pub.10.1007/s00210-007-0204-4

0 references

Structure-activity relationships of histamine H2 receptor ligands

1 reference

https://api.crossref.org/works/10.1007%2FS00210-007-0204-4

21 January 2018

The enzymatic preparation of [α-32P]nucleoside triphosphates, cyclic [32P]AMP, and cyclic [32P]GMP

1 reference

https://api.crossref.org/works/10.1007%2FS00210-007-0204-4

21 January 2018

Molecular mechanisms of ligand binding, signaling, and regulation within the superfamily of G-protein-coupled receptors: molecular modeling and mutagenesis approaches to receptor structure and function

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Distinct interaction of human and guinea pig histamine H2-receptor with guanidine-type agonists.

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Expression of Gs alpha in Escherichia coli. Purification and properties of two forms of the protein.

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The human histamine H2-receptor couples more efficiently to Sf9 insect cell Gs-proteins than to insect cell Gq-proteins: limitations of Sf9 cells for the analysis of receptor/Gq-protein coupling

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Synthesis and in vitro pharmacology of arpromidine and related phenyl(pyridylalkyl)guanidines, a potential new class of positive inotropic drugs

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Multiple residues in the second extracellular loop are critical for M3 muscarinic acetylcholine receptor activation

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Role of the second extracellular loop of adenosine receptors in agonist and antagonist binding. Analysis of chimeric A1/A3 adenosine receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Molecular basis for the interaction of histamine with the histamine H2 receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Mutations of Cys-17 and Ala-271 in the human histamine H2 receptor determine the species selectivity of guanidine-type agonists and increase constitutive activity

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The guinea pig histamine H2 receptor: gene cloning, tissue expression and chromosomal localization of its human counterpart

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Similar apparent constitutive activity of human histamine H(2)-receptor fused to long and short splice variants of G(salpha).

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Reconstitution of beta2-adrenoceptor-GTP-binding-protein interaction in Sf9 cells--high coupling efficiency in a beta2-adrenoceptor-G(s alpha) fusion protein

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Glutamate residues in the second extracellular loop of the human A2a adenosine receptor are required for ligand recognition

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Molecular cloning of the human histamine H2 receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The histamine H2 receptor agonist impromidine: synthesis and structure-activity considerations

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Oligomer formation of histamine H2 receptors expressed in Sf9 and COS7 cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identification of critical extracellular loop residues involved in alpha 1-adrenergic receptor subtype-selective antagonist binding

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Crystal structure of rhodopsin: A G protein-coupled receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

N1-(3-cyclohexylbutanoyl)-N2-[3-(1H-imidazol-4-yl)propyl]guanidine (UR-AK57), a potent partial agonist for the human histamine H1- and H2-receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Insights into ligand pharmacology using receptor-G-protein fusion proteins

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

International Union of Pharmacology. XIII. Classification of histamine receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Impromidine (SK&F 92676) is a very potent and specific agonist for histamine H2 receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

International Union of Pharmacology. XLVI. G protein-coupled receptor list.

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Probing ligand-specific histamine H1- and H2-receptor conformations with NG-acylated Imidazolylpropylguanidines

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Coupling of canine serotonin 5-HT(1B) and 5-HT(1D) receptor subtypes to the formation of inositol phosphates by dual interactions with endogenous G(i/o) and recombinant G(alpha15) proteins.

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Conformational changes of G protein-coupled receptors during their activation by agonist binding

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The second extracellular loop of the dopamine D2 receptor lines the binding-site crevice

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The agonistic binding site at the histamine H2 receptor. II. Theoretical investigations of histamine binding to receptor models of the seven alpha-helical transmembrane domain

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The binding site of aminergic G protein-coupled receptors: the transmembrane segments and second extracellular loop

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

GPCR-Galpha fusion proteins: molecular analysis of receptor-G-protein coupling

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Functional role of internal water molecules in rhodopsin revealed by X-ray crystallography.

1 reference

https://pubmed.ncbi.nlm.nih.gov/17999052

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1007/S00210-007-0204-4

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

16 September 2017

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