(Q43026301)

12 November 2017

title

Synthesis, 3D-QSAR, and structural modeling of benzolactam derivatives with binding affinity for the D(2) and D(3) receptors (English)

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12 November 2017

9

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12 November 2017

Eduardo Domínguez

5

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Christian F Masaguer

Christian F Masaguer

4

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Jana Selent

Jana Selent

2

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Jose Brea

José Brea

7

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Manuel Pastor

Manuel Pastor

10

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author name string

Laura López

1

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12 November 2017

Raquel Ortega

3

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12 November 2017

Filipe Areias

6

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12 November 2017

María Isabel Loza

8

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12 November 2017

language of work or name

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1 August 2010

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12 November 2017

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12 November 2017

volume

5

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12 November 2017

issue

8

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12 November 2017

page(s)

1300-1317

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Mesolimbic dopamine D3 receptors and use of antipsychotics in patients with schizophrenia. A postmortem study.

12 November 2017

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S33138 (N-[4-[2-[(3aS,9bR)-8-cyano-1,3a,4,9b-tetrahydro[1] benzopyrano[3,4-c]pyrrol-2(3H)-yl)-ethyl]phenyl-acetamide), a preferential dopamine D3 versus D2 receptor antagonist and potential antipsychotic agent: III. Actions in models of therapeutic

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Synthesis, binding affinity and SAR of new benzolactam derivatives as dopamine D3 receptor ligands

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Development of novel 1,2,3,4-tetrahydroisoquinoline derivatives and closely related compounds as potent and selective dopamine D3 receptor ligands

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Beta(1)-selective agonist (-)-1-(3,4-dimethoxyphenetylamino)-3-(3,4-dihydroxy)-2-propanol [(-)-RO363] differentially interacts with key amino acids responsible for beta(1)-selective binding in resting and active states

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Synthesis and pharmacological screening of some N-(4-substituted-piperazin-1-ylalkyl)-3,4-pyrroledicarboximides

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Synthesis and structure-activity relationships of new arylpiperazines: para substitution with electron-withdrawing groups decrease binding to 5-HT(1A) and D(2A) receptors

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7 January 2021

Identifiers

DOI

10.1002/CMDC.201000101

1 reference

12 November 2017

1 reference