(Q34503961)

2 August 2017

title

Target engagement and drug residence time can be observed in living cells with BRET. (English)

1 reference

2 August 2017

Matthew B Robers

1

1 reference

2 August 2017

Melanie L Dart

2

1 reference

2 August 2017

Carolyn C Woodroofe

3

1 reference

2 August 2017

Chad A Zimprich

4

1 reference

2 August 2017

Thomas A Kirkland

5

1 reference

2 August 2017

Thomas Machleidt

6

1 reference

2 August 2017

Kevin R Kupcho

7

1 reference

2 August 2017

Sergiy Levin

8

1 reference

2 August 2017

James R Hartnett

9

1 reference

2 August 2017

Kristopher Zimmerman

10

1 reference

2 August 2017

Andrew L Niles

11

1 reference

2 August 2017

Rachel Friedman Ohana

12

1 reference

2 August 2017

Danette L Daniels

13

1 reference

2 August 2017

Michael Slater

14

1 reference

2 August 2017

Monika G Wood

15

1 reference

2 August 2017

Mei Cong

16

1 reference

2 August 2017

Yi-Qiang Cheng

17

1 reference

2 August 2017

Keith V Wood

18

1 reference

2 August 2017

language of work or name

English

0 references

publication date

3 December 2015

1 reference

2 August 2017

published in

Nature Communications

1 reference

2 August 2017

volume

6

1 reference

2 August 2017

page(s)

10091

1 reference

Creative Commons Attribution 4.0 International

2 August 2017

copyright license

start time

1 December 2015

1 reference

April 2022 Public Data File from Crossref

copyright status

copyrighted

0 references

exact match

https://scigraph.springernature.com/pub.10.1038/ncomms10091

0 references

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7 July 2018

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7 July 2018

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7 July 2018

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7 July 2018

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7 July 2018

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7 July 2018

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7 July 2018

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7 July 2018

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7 July 2018

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Chemoproteomics reveals time-dependent binding of histone deacetylase inhibitors to endogenous repressor complexes.

7 July 2018

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Direct comparison of bioluminescence-based resonance energy transfer methods for monitoring of proteolytic cleavage

21 January 2018

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Characterization of the two catalytic domains in histone deacetylase 6.

21 January 2018

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HTS reporter displacement assay for fragment screening and fragment evolution toward leads with optimized binding kinetics, binding selectivity, and thermodynamic signature

21 January 2018

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Structural basis for the design and synthesis of selective HDAC inhibitors.

21 January 2018

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MGCD0103, a novel isotype-selective histone deacetylase inhibitor, has broad spectrum antitumor activity in vitro and in vivo

21 January 2018

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Direct comparison of fluorescence- and bioluminescence-based resonance energy transfer methods for real-time monitoring of thrombin-catalysed proteolytic cleavage

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Bioluminescence resonance energy transfer (BRET) for the real-time detection of protein-protein interactions

27 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/26631872

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Toward selective histone deacetylase inhibitor design: homology modeling, docking studies, and molecular dynamics simulations of human class I histone deacetylases

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/26631872

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1038/NCOMMS10091

1 reference

Dimensions Publication ID

2 August 2017

0 references

0 references

1 reference

2 August 2017

1 reference