(Q37011508)

17 August 2017

Sekikaic acid and lobaric acid target a dynamic interface of the coactivator CBP/p300. (English)

1 reference

17 August 2017

1 reference

1 reference

Giselle Tamayo-Castillo

11

1 reference

17 August 2017

Jonas W Højfeldt

2

0 references

author name string

Chinmay Y Majmudar

1

1 reference

17 August 2017

Carl J Arevang

3

1 reference

17 August 2017

William C Pomerantz

4

1 reference

17 August 2017

Jessica K Gagnon

5

1 reference

17 August 2017

Pamela J Schultz

6

1 reference

17 August 2017

Laura C Cesa

7

1 reference

17 August 2017

Conor H Doss

8

1 reference

17 August 2017

Steven P Rowe

9

1 reference

17 August 2017

Victor Vásquez

10

1 reference

17 August 2017

Tomasz Cierpicki

12

1 reference

17 August 2017

Charles L Brooks

13

1 reference

17 August 2017

David H Sherman

14

1 reference

17 August 2017

Anna K Mapp

15

1 reference

17 August 2017

language of work or name

English

0 references

publication date

8 October 2012

1 reference

full work available at URL

17 August 2017

https://europepmc.org/articles/pmc3711073?pdf=render

1 reference

19 March 2024

https://api.unpaywall.org/v2/10.1002/anie.201206815?email=unpaywall_01@example.com

published in

Angewandte Chemie International Edition

0 references

volume

51

1 reference

17 August 2017

45

1 reference

17 August 2017

11258-11262

1 reference

https://api.unpaywall.org/v2/10.1002/anie.201206815?email=unpaywall_01@example.com

17 August 2017

1 reference

19 March 2024

access restriction status

open access

1 reference

inferred from online access status

cites work

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Direct and selective small-molecule activation of proapoptotic BAX

29 September 2017

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Comparison of tertiary structures of proteins in protein-protein complexes with unbound forms suggests prevalence of allostery in signalling proteins.

29 September 2017

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Conformational control of the binding of the transactivation domain of the MLL protein and c-Myb to the KIX domain of CREB

29 September 2017

1 reference

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Small-molecule stabilization of protein-protein interactions: an underestimated concept in drug discovery?

29 September 2017

1 reference

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Caught in the act: covalent cross-linking captures activator-coactivator interactions in vivo.

29 September 2017

1 reference

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Thermodynamics-based drug design: strategies for inhibiting protein-protein interactions

29 September 2017

1 reference

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The role of CREB signaling in Alzheimer's disease and other cognitive disorders.

29 September 2017

1 reference

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Transient-state kinetic analysis of transcriptional activator·DNA complexes interacting with a key coactivator

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Leu628 of the KIX domain of CBP is a key residue for the interaction with the MLL transactivation domain

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Allosteric regulation of protease activity by small molecules.

29 September 2017

1 reference

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Disrupting protein-protein interactions with non-peptidic, small molecule alpha-helix mimetics

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Transcriptional switches: chemical approaches to gene regulation

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Discovery of a small-molecule inhibitor of the KIX-KID interaction

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

A high-resolution interaction map of three transcriptional activation domains with a key coactivator from photo-cross-linking and multiplexed mass spectrometry

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Tra1 as a screening target for transcriptional activation domain discovery

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Direct observation of the dynamic process underlying allosteric signal transmission.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Inhibition of transcription factors with small organic molecules

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Four domains of p300 each bind tightly to a sequence spanning both transactivation subdomains of p53

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Isolation and characterization of coactivator-binding peptoids from a combinatorial library

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

A transcription factor-binding domain of the coactivator CBP is essential for long-term memory and the expression of specific target genes

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Small molecule modulators of transcription

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Targets of the Gal4 transcription activator in functional transcription complexes.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Chemical approaches to transcriptional regulation

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Function of a eukaryotic transcription activator during the transcription cycle

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Intrinsically unstructured proteins and their functions

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Identification of small-molecule antagonists that inhibit an activator: coactivator interaction

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Small-molecule inhibitors of protein-protein interactions: progressing towards the dream

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

A wrench-shaped synthetic molecule that modulates a transcription factor-coactivator interaction.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Molecular Recognition of Protein Surfaces: High Affinity Ligands for the CBP KIX Domain

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Cooperativity in transcription factor binding to the coactivator CREB-binding protein (CBP). The mixed lineage leukemia protein (MLL) activation domain binds to an allosteric site on the KIX domain

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Pharmaceutically relevant metabolites from lichens

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Minimal activators that bind to the KIX domain of p300/CBP identified by phage display screening

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

CBP/p300 in cell growth, transformation, and development

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

A transcriptional activating region with two contrasting modes of protein interaction

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Solution Structure of the KIX Domain of CBP Bound to the Transactivation Domain of CREB: A Model for Activator:Coactivator Interactions

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Transcriptional activation by recruitment

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

A novel ring-expanded product with enhanced tyrosinase inhibitory activity from classical Fe-catalyzed oxidation of rosmarinic acid, a potent antioxidative Lamiaceae polyphenol

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Transcriptional tools: Small molecules for modulating CBP KIX-dependent transcriptional activators

27 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Impact of nonnatural amino acid mutagenesis on the in vivo function and binding modes of a transcriptional activator

27 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Amphipathic small molecules mimic the binding mode and function of endogenous transcription factors

27 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Systematic in vivo structure-function analysis of p300 in hematopoiesis

27 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Natural product inhibitors of protein-protein interactions mediated by Src-family SH2 domains.

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Allosteric switches: remote controls for proteins.

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Differential role for CBP and p300 CREB-binding domain in motor skill learning.

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Mechanism of transcription factor recruitment by acidic activators.

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Solution structure of the KIX domain of CBP bound to the transactivation domain of c-Myb

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Linking transcriptional mediators via the GACKIX domain super family.

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Structurally distinct modes of recognition of the KIX domain of CBP by Jun and CREB.

4 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3711073

Structural Basis for Cooperative Transcription Factor Binding to the CBP Coactivator

4 September 2018

1 reference

Crossref

https://api.crossref.org/works/10.1002%2FANIE.201206815

Structural analyses of CREB-CBP transcriptional activator-coactivator complexes by NMR spectroscopy: implications for mapping the boundaries of structural domains

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1002%2FANIE.201206815

Converting inactive peptides into potent transcriptional activators

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23042634

12 December 2020

inferred from PubMed ID database lookup

Antioxidant activity of some lichen metabolites

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23042634

12 December 2020

inferred from PubMed ID database lookup

How transcriptional activators bind target proteins

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23042634

12 December 2020

inferred from PubMed ID database lookup

Identifiers

DOI

10.1002/ANIE.201206815

1 reference

17 August 2017

1 reference

17 August 2017

PubMed publication ID

23042634

1 reference