(Q27690221)

10

0 references

Hans Wienk

9

0 references

Luc Brunsveld

object named as

Luc Brunsveld

13

0 references

Marcel Scheepstra

object named as

Marcel Scheepstra

1

0 references

Lech-Gustav Milroy

12

object named as

Lech-Gustav Milroy

0 references

author name string

Lidia Nieto

2

0 references

Anna K H Hirsch

3

0 references

Sascha Fuchs

4

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Seppe Leysen

5

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Chan Vinh Lam

6

0 references

Leslie in het Panhuis

7

0 references

Constant A A van Boeckel

Angewandte Chemie International Edition

8

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language of work or name

English

0 references

publication date

16 June 2014

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published in

0 references

volume

53

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issue

25

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page(s)

6443-8

0 references

cites work

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Ordering a Dynamic Protein Via a Small-Molecule Stabilizer

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Structural overview of the nuclear receptor superfamily: insights into physiology and therapeutics

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Mechanism of the nuclear receptor molecular switch

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The nuclear receptor superfamily and drug discovery

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Minireview: Not picking pockets: nuclear receptor alternate-site modulators (NRAMs)

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Antidiabetic actions of a non-agonist PPARγ ligand blocking Cdk5-mediated phosphorylation

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Noncanonical mechanisms to regulate nuclear receptor signaling

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Coregulator function: a key to understanding tissue specificity of selective receptor modulators

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Novel selective inhibitors of the interaction of individual nuclear hormone receptors with a mutually shared steroid receptor coactivator 2.

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Design and structure of stapled peptides binding to estrogen receptors

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Inhibition of α-helix-mediated protein-protein interactions using designed molecules

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Discovery of small molecule inhibitors of the interaction of the thyroid hormone receptor with transcriptional coregulators

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Inhibitors of the interaction of a thyroid hormone receptor and coactivators: preliminary structure-activity relationships.

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Alternative inhibition of androgen receptor signaling: peptidomimetic pyrimidines as direct androgen receptor/coactivator disruptors

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Discovery of the first irreversible small molecule inhibitors of the interaction between the vitamin D receptor and coactivators

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Design, synthesis, and in vitro biological evaluation of small molecule inhibitors of estrogen receptor alpha coactivator binding

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A surface on the androgen receptor that allosterically regulates coactivator binding

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Discovering small-molecule estrogen receptor α/coactivator binding inhibitors: high-throughput screening, ligand development, and models for enhanced potency

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"True" antiandrogens-selective non-ligand-binding pocket disruptors of androgen receptor-coactivator interactions: novel tools for prostate cancer

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Synthesis and biological evaluation of guanylhydrazone coactivator binding inhibitors for the estrogen receptor

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Natural-product-derived fragments for fragment-based ligand discovery

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Design of selective nuclear receptor modulators: RAR and RXR as a case study

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Complete relaxation and conformational exchange matrix (CORCEMA) analysis of intermolecular saturation transfer effects in reversibly forming ligand-receptor complexes

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Quantitative Analysis of STD-NMR Spectra of Reversibly Forming Ligand-Receptor Complexes.

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Triterpenoids and rexinoids as multifunctional agents for the prevention and treatment of cancer.

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RAR and RXR modulation in cancer and metabolic disease

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ApoE-directed therapeutics rapidly clear β-amyloid and reverse deficits in AD mouse models

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Synthetic retinoids: structure-activity relationships

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Identification of a naturally occurring rexinoid, honokiol, that activates the retinoid X receptor

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Honokiol increases ABCA1 expression level by activating retinoid X receptor beta.

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Therapeutic applications of compounds in the Magnolia family

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The natural product honokiol inhibits calcineurin inhibitor-induced and Ras-mediated tumor promoting pathways

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Honokiol inhibits non-small cell lung cancer cell migration by targeting PGE₂-mediated activation of β-catenin signaling

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Honokiol analogs: a novel class of anticancer agents targeting cell signaling pathways and other bioactivities.

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The rise of fragment-based drug discovery

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The combinatorial synthesis of bicyclic privileged structures or privileged substructures.

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Nuclear receptor-coregulator interaction profiling identifies TRIP3 as a novel peroxisome proliferator-activated receptor gamma cofactor

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Ligand efficiency indices for effective drug discovery

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A detergent-based assay for the detection of promiscuous inhibitors

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Modulators of the structural dynamics of the retinoid X receptor to reveal receptor function

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Palladium-Catalyzed Borylation of Aryl Chlorides: Scope, Applications, and Computational Studies

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