(Q34297570)

1 August 2017

title

The allosteric vestibule of a seven transmembrane helical receptor controls G-protein coupling (English)

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1 August 2017

main subject

transmembrane protein

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8

Carlo Matera

1 reference

1 August 2017

Andreas Bock

1

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Clelia Dallanoce

object named as

Clelia Dallanoce

4

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Marco De Amici

object named as

Marco De Amici

16

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Ulrike Holzgrabe

object named as

Ulrike Holzgrabe

17

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author name string

Nicole Merten

2

1 reference

1 August 2017

Ramona Schrage

3

1 reference

1 August 2017

Julia Bätz

5

1 reference

1 August 2017

Jessica Klöckner

6

1 reference

1 August 2017

Jens Schmitz

7

1 reference

1 August 2017

Katharina Simon

9

1 reference

1 August 2017

Anna Kebig

10

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1 August 2017

Lucas Peters

11

1 reference

1 August 2017

Anke Müller

12

1 reference

1 August 2017

Jasmin Schrobang-Ley

13

1 reference

1 August 2017

Christian Tränkle

14

1 reference

1 August 2017

Carsten Hoffmann

15

1 reference

1 August 2017

Evi Kostenis

18

1 reference

1 August 2017

Klaus Mohr

19

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1 August 2017

language of work or name

English

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publication date

1 January 2012

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1 August 2017

published in

Nature Communications

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1 August 2017

volume

3

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1 August 2017

page(s)

1044

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Creative Commons Attribution-NonCommercial-NoDerivs 3.0 Unported

1 August 2017

copyright license

start time

1 January 2012

1 reference

April 2022 Public Data File from Crossref

copyright status

copyrighted

0 references

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6 July 2018

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6 July 2018

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The C-terminal tail of CRTH2 is a key molecular determinant that constrains Galphai and downstream signaling cascade activation

6 July 2018

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Dualsteric GPCR targeting: a novel route to binding and signaling pathway selectivity

6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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Operational models of pharmacological agonism.

6 July 2018

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6 July 2018

1 reference

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Diversity of G proteins in signal transduction

6 July 2018

1 reference

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Applying label-free dynamic mass redistribution technology to frame signaling of G protein-coupled receptors noninvasively in living cells.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3658004

Deconvolution of complex G protein-coupled receptor signaling in live cells using dynamic mass redistribution measurements.

28 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3658004

Allosteric small molecules unveil a role of an extracellular E2/transmembrane helix 7 junction for G protein-coupled receptor activation

28 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3658004

Allosteric Modulation of G Protein–Coupled Receptors

28 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3658004

Critical amino acid residues of the common allosteric site on the M2 muscarinic acetylcholine receptor: more similarities than differences between the structurally divergent agents gallamine and bis(ammonio)alkane-type hexamethylene-bis-[dimethyl-(3

28 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3658004

Interactions of orthosteric and allosteric ligands with [3H]dimethyl-W84 at the common allosteric site of muscarinic M2 receptors

28 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3658004

Allosteric site on muscarinic acetylcholine receptors: identification of two amino acids in the muscarinic M2 receptor that account entirely for the M2/M5 subtype selectivities of some structurally diverse allosteric ligands in N-methylscopolamine-o

28 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3658004

Measurement of the millisecond activation switch of G protein-coupled receptors in living cells

28 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3658004

Inhibition of the actions of carbachol and DFP on guinea pig isolated atria by alkane-bis-ammonium compounds

28 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3658004

Linkage of G protein-coupled receptors to the MAPK signaling pathway through PI 3-kinase gamma

28 October 2018

1 reference

12 December 2020

Allosteric interactions with muscarinic acetylcholine receptors: complex role of the conserved tryptophan M2422Trp in a critical cluster of amino acids for baseline affinity, subtype selectivity, and cooperativity

1 reference

12 December 2020

Modification of the binding properties of muscarinic receptors by gallamine

1 reference

12 December 2020

Agonist-independent inhibition of G protein activation by muscarinic acetylcholine receptor antagonists in cardiac membranes

1 reference

12 December 2020

Convergent, short synthesis of the muscarinic superagonist iperoxo

1 reference

Crossref

https://api.crossref.org/works/10.1038%2FNCOMMS2028

7 January 2021

inferred from DOI database lookup

Identifiers

DOI

10.1038/NCOMMS2028

1 reference

Dimensions Publication ID

1 August 2017

0 references

0 references

1 reference

1 August 2017

1 reference