(Q37789790)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20849671%20AND%20SRC:MED&resulttype=core&format=json

14 February 2020

title

The structural basis of function in Cys-loop receptors (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20849671%20AND%20SRC:MED&resulttype=core&format=json

14 February 2020

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20849671%20AND%20SRC:MED&resulttype=core&format=json

14 February 2020

3

Sarah C R Lummis

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20849671%20AND%20SRC:MED&resulttype=core&format=json

14 February 2020

author name string

Andrew J Thompson

series ordinal

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20849671%20AND%20SRC:MED&resulttype=core&format=json

14 February 2020

publication date

20 September 2010

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20849671%20AND%20SRC:MED&resulttype=core&format=json

Quarterly Reviews of Biophysics

14 February 2020

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20849671%20AND%20SRC:MED&resulttype=core&format=json

14 February 2020

volume

43

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20849671%20AND%20SRC:MED&resulttype=core&format=json

14 February 2020

issue

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20849671%20AND%20SRC:MED&resulttype=core&format=json

14 February 2020

page(s)

449-499

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20849671%20AND%20SRC:MED&resulttype=core&format=json

Ion permeation and conduction in a human recombinant 5-HT3 receptor subunit (h5-HT3A).

14 February 2020

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Identification of channel-lining residues in the M2 membrane-spanning segment of the GABA(A) receptor alpha1 subunit

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Nicotine binding to brain receptors requires a strong cation-pi interaction

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A unified view of the role of electrostatic interactions in modulating the gating of Cys loop receptors

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21 January 2018

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A conserved cysteine residue in the third transmembrane domain is essential for homomeric 5-HT3 receptor function

21 January 2018

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Mutations at the GABA receptor selectivity filter: a possible role for effective charges

21 January 2018

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Mutations at two distinct sites within the channel domain M2 alter calcium permeability of neuronal alpha 7 nicotinic receptor

21 January 2018

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The intrinsic electrostatic potential and the intermediate ring of charge in the acetylcholine receptor channel

21 January 2018

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On the Benzodiazepine Binding Pocket in GABAA Receptors

21 January 2018

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Acetylcholine receptor channel structure in the resting, open, and desensitized states probed with the substituted-cysteine-accessibility method

21 January 2018

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GABA(A) receptor M2-M3 loop secondary structure and changes in accessibility during channel gating.

21 January 2018

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The location of the gate in the acetylcholine receptor channel

21 January 2018

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EXP-1 is an excitatory GABA-gated cation channel

21 January 2018

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Gamma-aminobutyric acid increases the water accessibility of M3 membrane-spanning segment residues in gamma-aminobutyric acid type A receptors

21 January 2018

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Tyrosine residues that control binding and gating in the 5-hydroxytryptamine3 receptor revealed by unnatural amino acid mutagenesis.

21 January 2018

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Organization of the mouse 5-HT3 receptor gene and functional expression of two splice variants

21 January 2018

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Cation-pi interactions in ligand recognition by serotonergic (5-HT3A) and nicotinic acetylcholine receptors: the anomalous binding properties of nicotine

21 January 2018

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Cyclic AMP-dependent protein kinase (PKA) and protein kinase C phosphorylate sites in the amino acid sequence corresponding to the M3/M4 cytoplasmic domain of alpha4 neuronal nicotinic receptor subunits

21 January 2018

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Molecular pharmacology of the glycine receptor chloride channel

21 January 2018

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The activation mechanism of alpha1 homomeric glycine receptors

21 January 2018

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Establishing an ion pair interaction in the homomeric rho1 gamma-aminobutyric acid type A receptor that contributes to the gating pathway.

21 January 2018

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First genetic evidence of GABA(A) receptor dysfunction in epilepsy: a mutation in the gamma2-subunit gene

21 January 2018

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Structural basis of activation of cys-loop receptors: the extracellular-transmembrane interface as a coupling region

21 January 2018

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X-ray structure of a pentameric ligand-gated ion channel in an apparently open conformation

21 January 2018

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Atomic force microscopy reveals the stoichiometry and subunit arrangement of 5-HT3 receptors

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Modulation of the expression of GABA(A) receptors in rat cerebellar granule cells by protein tyrosine kinases and protein kinase C.

21 January 2018

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Toward biophysical probes for the 5-HT3 receptor: structure-activity relationship study of granisetron derivatives

21 January 2018

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Gating at the mouth of the acetylcholine receptor channel: energetic consequences of mutations in the alphaM2-cap

21 January 2018

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Identification of critical residues in loop E in the 5-HT3ASR binding site

21 January 2018

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Fourier transform infrared and hydrogen/deuterium exchange reveal an exchange-resistant core of alpha-helical peptide hydrogens in the nicotinic acetylcholine receptor.

21 January 2018

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Functional group interactions of a 5-HT3R antagonist

21 January 2018

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SR 57227A: a potent and selective agonist at central and peripheral 5-HT3 receptors in vitro and in vivo.

21 January 2018

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Genetic and biochemical evidence for a novel avermectin-sensitive chloride channel in Caenorhabditis elegans. Isolation and characterization.

21 January 2018

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Anesthetics as chemical tools to study the structure and function of nicotinic acetylcholine receptors

21 January 2018

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Identification of two novel Drosophila melanogaster histamine-gated chloride channel subunits expressed in the eye.

21 January 2018

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Potentials of mean force for acetylcholine unbinding from the alpha7 nicotinic acetylcholine receptor ligand-binding domain

21 January 2018

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Volatile general anaesthetic actions on recombinant nACh alpha 7, 5-HT3 and chimeric nACh alpha 7-5-HT3 receptors expressed in Xenopus oocytes

21 January 2018

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Contribution of the beta subunit M2 segment to the ion-conducting pathway of the acetylcholine receptor

21 January 2018

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Identification of acetylcholine receptor channel-lining residues in the M1 segment of the beta-subunit.

21 January 2018

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Ca2+ ions block and permeate serotonin 5-HT3 receptor channels in rat hippocampal interneurons

21 January 2018

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A sequence in the main cytoplasmic loop of the alpha subunit is required for assembly of mouse muscle nicotinic acetylcholine receptor

21 January 2018

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Interactions of anesthetics with their targets: non-specific, specific or both?

21 January 2018

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Structural elements near the C-terminus are responsible for changes in nicotinic receptor gating kinetics following patch excision

21 January 2018

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Activation of the nicotinic acetylcholine receptor involves a switch in conformation of the alpha subunits.

21 January 2018

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Identification of acetylcholine receptor channel-lining residues in the entire M2 segment of the alpha subunit.

21 January 2018

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Refined structure of the nicotinic acetylcholine receptor at 4A resolution

21 January 2018

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Acetylcholine receptor channel structure probed in cysteine-substitution mutants.

21 January 2018

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The Croonian Lecture 2000. Nicotinic acetylcholine receptor and the structural basis of fast synaptic transmission

21 January 2018

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Identification of acetylcholine receptor channel-lining residues in the M1 segment of the alpha-subunit.

21 January 2018

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Pore structure of the Cys-loop ligand-gated ion channels

21 January 2018

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A molecular basis for agonist and antagonist actions at GABA(C) receptors

21 January 2018

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Tissue-specific alternative promoters of the serotonin receptor gene HTR3B in human brain and intestine.

21 January 2018

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Comparative modeling of a GABAA alpha1 receptor using three crystal structures as templates

21 January 2018

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Modeling noncompetitive antagonism of a nicotinic acetylcholine receptor

21 January 2018

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Loop B is a major structural component of the 5-HT3 receptor.

21 January 2018

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Mutagenesis and molecular modeling reveal the importance of the 5-HT3 receptor F-loop

21 January 2018

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Unbinding pathways of an agonist and an antagonist from the 5-HT3 receptor

21 January 2018

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Locating an antagonist in the 5-HT3 receptor binding site using modeling and radioligand binding.

21 January 2018

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Antimalarial drugs inhibit human 5-HT(3) and GABA(A) but not GABA(C) receptors

21 January 2018

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Calcium modulation of 5-HT3 receptor binding and function

21 January 2018

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https://api.crossref.org/works/10.1017%2FS0033583510000168

In pursuit of the high-resolution structure of nicotinic acetylcholine receptors

21 January 2018

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21 January 2018

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A single ring of charged amino acids at one end of the pore can control ion selectivity in the 5-HT3 receptor

21 January 2018

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Ca2+ permeability of the (alpha4)3(beta2)2 stoichiometry greatly exceeds that of (alpha4)2(beta2)3 human acetylcholine receptors.

21 January 2018

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Two neighboring residues of loop A of the alpha1 subunit point towards the benzodiazepine binding site of GABAA receptors

21 January 2018

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Functional effects of periodic tryptophan substitutions in the alpha M4 transmembrane domain of the Torpedo californica nicotinic acetylcholine receptor

21 January 2018

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Alteration in ion channel function of mouse nicotinic acetylcholine receptor by mutations in the M4 transmembrane domain

21 January 2018

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The diverse actions of volatile and gaseous anesthetics on human-cloned 5-hydroxytryptamine3 receptors expressed in Xenopus oocytes

21 January 2018

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The loop C region of the murine 5-HT3A receptor contributes to the differential actions of 5-hydroxytryptamine and m-chlorophenylbiguanide

21 January 2018

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Modulation of 5-HT3 receptor-mediated response and trafficking by activation of protein kinase C.

21 January 2018

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https://api.crossref.org/works/10.1017%2FS0033583510000168

Defining the roles of Asn-128, Glu-129 and Phe-130 in loop A of the 5-HT3 receptor

21 January 2018

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Mechanistic contributions of residues in the M1 transmembrane domain of the nicotinic receptor to channel gating

21 January 2018

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The role of tryptophan residues in the 5-Hydroxytryptamine(3) receptor ligand binding domain

21 January 2018

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Gating of nicotinic ACh receptors: latest insights into ligand binding and function

21 January 2018

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The pore dimensions of gramicidin A.

21 January 2018

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Codon optimization of Caenorhabditis elegans GluCl ion channel genes for mammalian cells dramatically improves expression levels.

21 January 2018

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The molecular basis of the structure and function of the 5-HT3 receptor: a model ligand-gated ion channel (review)

21 January 2018

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On the origin of ion selectivity in the Cys-loop receptor family

21 January 2018

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Number and locations of agonist binding sites required to activate homomeric Cys-loop receptors

21 January 2018

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MOD-1 is a serotonin-gated chloride channel that modulates locomotory behaviour in C. elegans

21 January 2018

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Mutation of an arginine residue in the human glycine receptor transforms beta-alanine and taurine from agonists into competitive antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Three putative N-glycosylation sites within the murine 5-HT3A receptor sequence affect plasma membrane targeting, ligand binding, and calcium influx in heterologous mammalian cells

21 January 2018

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A stepwise mechanism for acetylcholine receptor channel gating

21 January 2018

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https://api.crossref.org/works/10.1017%2FS0033583510000168

A hydrogen bond in loop A is critical for the binding and function of the 5-HT3 receptor.

21 January 2018

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https://api.crossref.org/works/10.1017%2FS0033583510000168

Illuminating the structure and function of Cys-loop receptors

21 January 2018

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https://api.crossref.org/works/10.1017%2FS0033583510000168

Role of the conserved lysine residue in the middle of the predicted extracellular loop between M2 and M3 in the GABA(A) receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The benzodiazepine binding site of GABAA receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Mapping of the benzodiazepine recognition site on GABA(A) receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

FUGUE: sequence-structure homology recognition using environment-specific substitution tables and structure-dependent gap penalties

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Functional stoichiometry at the nicotinic receptor. The photon cross section for phase 1 corresponds to two bis-Q molecules per channel

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Comparative surface accessibility of a pore-lining threonine residue (T6') in the glycine and GABA(A) receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A single beta subunit M2 domain residue controls the picrotoxin sensitivity of alphabeta heteromeric glycine receptor chloride channels

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A Mutation in Transmembrane Domain II of the 5-Hydroxytryptamine3A Receptor Stabilizes Channel Opening and Alters Alcohol Modulatory Actions

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A cation-pi interaction in the binding site of the glycine receptor is mediated by a phenylalanine residue

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Phosphorylation of the recombinant rho1 GABA receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Conformational variability of the glycine receptor M2 domain in response to activation by different agonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Distinct conformational changes in activated agonist-bound and agonist-free glycine receptor subunits

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Molecular determinants of single-channel conductance and ion selectivity in the Cys-loop family: insights from the 5-HT3 receptor.

21 January 2018

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https://api.crossref.org/works/10.1017%2FS0033583510000168

The 5-hydroxytryptamine type 3 (5-HT3) receptor reveals a novel determinant of single-channel conductance.

21 January 2018

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https://api.crossref.org/works/10.1017%2FS0033583510000168

Single-molecule imaging of a fluorescent unnatural amino acid incorporated into nicotinic receptors

21 January 2018

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https://api.crossref.org/works/10.1017%2FS0033583510000168

Minimal structural rearrangement of the cytoplasmic pore during activation of the 5-HT3A receptor

21 January 2018

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Novel structural determinants of single channel conductance and ion selectivity in 5-hydroxytryptamine type 3 and nicotinic acetylcholine receptors

21 January 2018

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Characterization of the ligand-binding site of the serotonin 5-HT3 receptor: the role of glutamate residues 97, 224, AND 235.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A highly conserved aspartic acid residue in the signature disulfide loop of the alpha 1 subunit is a determinant of gating in the glycine receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Structural model of nicotinic acetylcholine receptor isotypes bound to acetylcholine and nicotine

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Assembly of GABA(A) receptors (Review).

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The F-loop of the GABA A receptor gamma2 subunit contributes to benzodiazepine modulation

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Comparative protein modelling by satisfaction of spatial restraints

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Unnatural amino acid mutagenesis of the GABA(A) receptor binding site residues reveals a novel cation-pi interaction between GABA and beta 2Tyr97

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Mutations in the M4 domain of the Torpedo californica nicotinic acetylcholine receptor alter channel opening and closing

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Fishing for allosteric sites on GABA(A) receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

GABA A receptors: subtypes provide diversity of function and pharmacology

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Docking and scoring of metallo-beta-lactamases inhibitors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Arg-274 and Leu-277 of the gamma-aminobutyric acid type A receptor alpha 2 subunit define agonist efficacy and potency

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Crystal structure of the extracellular domain of a bacterial ligand-gated ion channel

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Primary structure of α-subunit precursor of Torpedo californica acetylcholine receptor deduced from cDNA sequence

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

On the voltage-dependent Ca2+ block of serotonin 5-HT3 receptors: a critical role of intracellular phosphates

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Cyanotriphenylborate: subtype-specific blocker of glycine receptor chloride channels

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

GABA(A) receptor subtypes: dissecting their pharmacological functions

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Gating of alpha3beta4 neuronal nicotinic receptor can be controlled by the loop M2-M3 of both alpha3 and beta4 subunits.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A residue in the middle of the M2-M3 loop of the beta4 subunit specifically affects gating of neuronal nicotinic receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Central nicotinic receptors: structure, function, ligands, and therapeutic potential.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

BUILDER v.2: improving the chemistry of a de novo design strategy

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Prediction of 5-HT3 receptor agonist-binding residues using homology modeling.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Effects of PKC and PKA phosphorylation on desensitization of nicotinic acetylcholine receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Structural and electrostatic properties of the 5-HT3 receptor pore revealed by substituted cysteine accessibility mutagenesis.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Activation of endogenous protein kinase C enhances currents through α1 and α2 glycine receptor channels

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Characterization of the novel human serotonin receptor subunits 5-HT3C,5-HT3D, and 5-HT3E

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Cloning, physical mapping and expression analysis of the human 5-HT3 serotonin receptor-like genes HTR3C, HTR3D and HTR3E.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The role of the agonist binding site in Ca(2+) inhibition of the recombinant 5-HT(3A) receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Nootropic alpha7 nicotinic receptor allosteric modulator derived from GABAA receptor modulators

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Charge scan reveals an extended region at the intracellular end of the GABA receptor pore that can influence ion selectivity

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Insights into the structural basis for zinc inhibition of the glycine receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Tryptophan substitutions reveal the role of nicotinic acetylcholine receptor alpha-TM3 domain in channel gating: differences between Torpedo and muscle-type AChR.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Response of acetylcholine receptors to photoisomerizations of bound agonist molecules

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Block by 5-hydroxytryptamine of neuronal acetylcholine receptor channels expressed in Xenopus oocytes.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Probing the role of backbone hydrogen bonding in a critical beta sheet of the extracellular domain of a cys-loop receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Local and global ligand-induced changes in the structure of the GABA(A) receptor.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Different binding orientations for the same agonist at homologous receptors: a lock and key or a simple wedge?

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Molecular characterisation of a pH-gated chloride channel from Sarcoptes scabiei.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

alpha4beta2 nicotinic receptors with high and low acetylcholine sensitivity: pharmacology, stoichiometry, and sensitivity to long-term exposure to nicotine.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Stoichiometry and pharmacology of two human alpha4beta2 nicotinic receptor types

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Single channel analysis of conductance and rectification in cation-selective, mutant glycine receptor channels

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Cloning, expression, and characterization of ferret 5-HT(3) receptor subunit

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Structure and gating mechanism of the acetylcholine receptor pore

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Nicotinic acetylcholine receptor at 4.6 A resolution: transverse tunnels in the channel wall.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Diversity of vertebrate nicotinic acetylcholine receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Flash decaging of tyrosine sidechains in an ion channel.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Assembly and trafficking of nicotinic acetylcholine receptors (Review).

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

RIC-3: a nicotinic acetylcholine receptor chaperone

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Secondary structure of the nicotinic acetylcholine receptor: implications for structural models of a ligand-gated ion channel.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Chimeric mutations in the M2 segment of the 5-hydroxytryptamine-gated chloride channel MOD-1 define a minimal determinant of anion/cation permeability

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Multifunctional basic motif in the glycine receptor intracellular domain induces subunit-specific sorting

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Molecular dynamics simulations of GABA binding to the GABAC receptor: the role of Arg104.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Physiological and pharmacological properties of 5-HT3 receptors — A patch clamp-study

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Binding interactions of antagonists with 5-hydroxytryptamine3A receptor models

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The 5-HT3 antagonist tropisetron (ICS 205-930) is a potent and selective alpha7 nicotinic receptor partial agonist

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Structure and dynamics of the second and third transmembrane domains of human glycine receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Drug interactions at GABA(A) receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Trafficking and synaptic anchoring of ionotropic inhibitory neurotransmitter receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Ligand-gated ion channels: mechanisms underlying ion selectivity

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Cation-selective mutations in the M2 domain of the inhibitory glycine receptor channel reveal determinants of ion-charge selectivity

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

M2 pore mutations convert the glycine receptor channel from being anion- to cation-selective

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A cytoplasmic region determines single-channel conductance in 5-HT3 receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Coupling of agonist binding to channel gating in the GABA(A) receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Charged Residues in the β2 Subunit Involved in GABAA Receptor Activation

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Identification of intracellular and extracellular domains mediating signal transduction in the inhibitory glycine receptor chloride channel

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Native glycine receptor subtypes and their physiological roles

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Molecular structure and function of the glycine receptor chloride channel

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Cis-trans isomerization at a proline opens the pore of a neurotransmitter-gated ion channel.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A cation-pi binding interaction with a tyrosine in the binding site of the GABAC receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Spatial structure of the M3 transmembrane segment of the nicotinic acetylcholine receptor alpha subunit

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Competitive antagonism between the nicotinic allosteric potentiating ligand galantamine and kynurenic acid at alpha7* nicotinic receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Agonists and antagonists bind to an A-A interface in the heteromeric 5-HT3AB receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Channel gating of the glycine receptor changes accessibility to residues implicated in receptor potentiation by alcohols and anesthetics

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Patch Clamp Study of Serotonin-Gated Currents via 5-HT Type 3 Receptors by Using a Novel Approach SHAM for Receptor Channel Scanning

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Interactions of granisetron with an agonist-free 5-HT3A receptor model

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Structural determinants of benzodiazepine allosteric regulation of GABA(A) receptor currents.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The beta subunit determines the ion selectivity of the GABAA receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Charge selectivity of the Cys-loop family of ligand-gated ion channels.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Mutational studies using a cation-conducting GABAA receptor reveal the selectivity determinants of the Cys-loop family of ligand-gated ion channels

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

3B but which 3B and that's just one of the questions: the heterogeneity of human 5-HT3 receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Modular design of Cys-loop ligand-gated ion channels: functional 5-HT3 and GABA rho1 receptors lacking the large cytoplasmic M3M4 loop

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Structural determinants of Ca2+ permeability and conduction in the human 5-hydroxytryptamine type 3A receptor.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Chemical scale studies of the Phe-Pro conserved motif in the cys loop of Cys loop receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Selective elimination of glutamate activation and introduction of fluorescent proteins into a Caenorhabditis elegans chloride channel

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Properties of human glycine receptors containing the hyperekplexia mutation alpha1(K276E), expressed in Xenopus oocytes.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The permeation pathway of neurotransmitter-gated ion channels

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Evidence that the M2 membrane-spanning region lines the ion channel pore of the nicotinic receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Conformation-dependent hydrophobic photolabeling of the nicotinic receptor: electrophysiology-coordinated photochemistry and mass spectrometry

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Principal pathway coupling agonist binding to channel gating in nicotinic receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Kinetics of unliganded acetylcholine receptor channel gating

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Binding to gating transduction in nicotinic receptors: Cys-loop energetically couples to pre-M1 and M2-M3 regions

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Spontaneous openings of the acetylcholine receptor channel

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Nicotinic receptor interloop proline anchors beta1-beta2 and Cys loops in coupling agonist binding to channel gating

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Noninvasive imaging of 5-HT3 receptor trafficking in live cells: from biosynthesis to endocytosis.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Water conduction through the hydrophobic channel of a carbon nanotube

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Functional differences between splice variants of the murine 5-HT(3A) receptor: possible role for phosphorylation

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Zn(2+) enhancement of the recombinant 5-HT(3) receptor is modulated by divalent cations

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Arginine 222 in the pre-transmembrane domain 1 of 5-HT3A receptors links agonist binding to channel gating

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The 5-HT3B subunit confers spontaneous channel opening and altered ligand properties of the 5-HT3 receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Mutations in the M4 domain of Torpedo californica acetylcholine receptor dramatically alter ion channel function

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Models of the extracellular domain of the nicotinic receptors and of agonist- and Ca2+-binding sites

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Tryptophan substitutions at the lipid-exposed transmembrane segment M4 of Torpedo californica acetylcholine receptor govern channel gating.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The properties of 5-HT3 receptors in clonal cell lines studied by patch-clamp techniques

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Channel gating governed symmetrically by conserved leucine residues in the M2 domain of nicotinic receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Role of aspartate 298 in mouse 5-HT3A receptor gating and modulation by extracellular Ca2+.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Zinc-mediated inhibition of GABA(A) receptors: discrete binding sites underlie subtype specificity

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Characterisation of 5-HT3C, 5-HT3D and 5-HT3E receptor subunits: evolution, distribution and function.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Nicotinic acetylcholine receptors: from structure to brain function

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Partial agonists as therapeutic agents at neuronal nicotinic acetylcholine receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

X-ray structure of a prokaryotic pentameric ligand-gated ion channel

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Structural determinants for interaction of partial agonists with acetylcholine binding protein and neuronal α7 nicotinic acetylcholine receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Structural mechanisms underlying benzodiazepine modulation of the GABA(A) receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Galanthamine and Non-competitive Inhibitor Binding to ACh-binding Protein: Evidence for a Binding Site on Non-α-subunit Interfaces of Heteromeric Neuronal Nicotinic Receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Structures of Aplysia AChBP complexes with nicotinic agonists and antagonists reveal distinctive binding interfaces and conformations

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Photochemical proteolysis of an unstructured linker of the GABAAR extracellular domain prevents GABA but not pentobarbital activation

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Common determinants of single channel conductance within the large cytoplasmic loop of 5-hydroxytryptamine type 3 and alpha4beta2 nicotinic acetylcholine receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

An intramembrane aromatic network determines pentameric assembly of Cys-loop receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Tryptophan scanning mutagenesis in the alphaM3 transmembrane domain of the Torpedo californica acetylcholine receptor: functional and structural implications

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Nicotinic agonists competitively antagonize serotonin at mouse 5-HT3 receptors expressed in Xenopus oocytes

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Conversion of the ion selectivity of the 5-HT(3a) receptor from cationic to anionic reveals a conserved feature of the ligand-gated ion channel superfamily

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A chimera encoding the fusion of an acetylcholine-binding protein to an ion channel is stabilized in a state close to the desensitized form of ligand-gated ion channels

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Molecular tuning of fast gating in pentameric ligand-gated ion channels

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Mapping the conformational wave of acetylcholine receptor channel gating

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The extracellular linker of muscle acetylcholine receptor channels is a gating control element

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Distinct profiles of alpha7 nAChR positive allosteric modulation revealed by structurally diverse chemotypes

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Mutation of the GABAA receptor M1 transmembrane proline increases GABA affinity and reduces barbiturate enhancement.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Expression of recombinant homo-oligomeric 5-hydroxytryptamine3 receptors provides new insights into their maturation and structure

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Distinct subcellular targeting of fluorescent nicotinic alpha 3 beta 4 and serotoninergic 5-HT3A receptors in hippocampal neurons

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Heterogeneity and complexity of native brain nicotinic receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Loose protein packing around the extracellular half of the GABA(A) receptor beta1 subunit M2 channel-lining segment

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

An electrophysiological investigation of the properties of a murine recombinant 5-HT3 receptor stably expressed in HEK 293 cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Gating of nicotinic ACh receptors; new insights into structural transitions triggered by agonist binding that induce channel opening

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Solution NMR of acetylcholine binding protein reveals agonist-mediated conformational change of the C-loop

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

"Optical patch-clamping": single-channel recording by imaging Ca2+ flux through individual muscle acetylcholine receptor channels

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Mutations in the channel domain of a neuronal nicotinic receptor convert ion selectivity from cationic to anionic.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Crystal structure of the extracellular domain of nAChR alpha1 bound to alpha-bungarotoxin at 1.94 A resolution

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Cation-pi interactions in structural biology

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Nicotinic receptor M3 transmembrane domain: position 8' contributes to channel gating

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The alphaM1 transmembrane segment of the nicotinic acetylcholine receptor interacts strongly with model membranes

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A novel class of ligand-gated ion channel is activated by Zn2+

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The 5-HT3B subunit is a major determinant of serotonin-receptor function

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A fluorophore attached to nicotinic acetylcholine receptor beta M2 detects productive binding of agonist to the alpha delta site

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The gating isomerization of neuromuscular acetylcholine receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Regulation of neuronal nicotinic receptor traffic and expression

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Cy3-3-acylcholine: a fluorescent analogue of acetylcholine for single molecule detection

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Alpha 4 beta 2 neuronal nicotinic acetylcholine receptors in the central nervous system are inhibited by isoflurane and propofol, but alpha 7-type nicotinic acetylcholine receptors are unaffected.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A histidine residue in the extracellular N-terminal domain of the GABA(A) receptor alpha5 subunit regulates sensitivity to inhibition by zinc

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Amphipathic analysis and possible formation of the ion channel in an acetylcholine receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Evidence that the TM1-TM2 loop contributes to the rho1 GABA receptor pore.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A lipid-dependent uncoupled conformation of the acetylcholine receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Probing ion-channel pores one proton at a time

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Pore-opening mechanism of the nicotinic acetylcholine receptor evinced by proton transfer

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Cloning of the gamma-aminobutyric acid (GABA) rho 1 cDNA: a GABA receptor subunit highly expressed in the retina

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

An amino acid substitution in the pore region of a glutamate-gated chloride channel enables the coupling of ligand binding to channel gating.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Cloning of an avermectin-sensitive glutamate-gated chloride channel from Caenorhabditis elegans

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Tryptophan substitutions at lipid-exposed positions of the gamma M3 transmembrane domain increase the macroscopic ionic current response of the Torpedo californica nicotinic acetylcholine receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Anxiety over GABA(A) receptor structure relieved by AChBP.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Enhancement of 5-hydroxytryptamine3A receptor function by phorbol 12-myristate, 13-acetate is mediated by protein kinase C and tyrosine kinase activity

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Atomic structure and dynamics of pentameric ligand-gated ion channels: new insight from bacterial homologues.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Allosteric modulators of the alpha7 nicotinic acetylcholine receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Protein interactions involving the gamma2 large cytoplasmic loop of GABA(A) receptors modulate conductance

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

GABAC receptor rho subunits are heterogeneously expressed in the human CNS and form homo- and heterooligomers with distinct physical properties

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Backbone mutations in transmembrane domains of a ligand-gated ion channel: implications for the mechanism of gating.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Point mutation in the first transmembrane region of the beta 2 subunit of the gamma--aminobutyric acid type A receptor alters desensitization kinetics of gamma--aminobutyric acid- and anesthetic-induced channel gating

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Native and cloned 5-HT(3A)(S) receptors are anchored to F-actin in clonal cells and neurons.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Chimaeric nicotinic-serotonergic receptor combines distinct ligand binding and channel specificities.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Single-channel kinetic analysis for activation and desensitization of homomeric 5-HT(3)A receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A kinetic mechanism for nicotinic acetylcholine receptors based on multiple allosteric transitions

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Trafficking of 5-HT(3) and GABA(A) receptors (Review).

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Mutations in M2 alter the selectivity of the mouse nicotinic acetylcholine receptor for organic and alkali metal cations

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

An open-channel blocker interacts with adjacent turns of α-helices in the nicotinic acetylcholine receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Acetylcholine receptor: an allosteric protein

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Allosteric activation mechanism of the cys-loop receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Site-specific fluorescence reveals distinct structural changes with GABA receptor activation and antagonism

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Glutamate 172, essential for modulation of L247T alpha7 ACh receptors by Ca2+, lines the extracellular vestibule

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Permeant but not impermeant divalent cations enhance activation of nondesensitizing alpha(7) nicotinic receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

An N-terminal histidine regulates Zn(2+) inhibition on the murine GABA(A) receptor beta3 subunit

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The pharmacological and functional characteristics of the serotonin 5-HT(3A) receptor are specifically modified by a 5-HT(3B) receptor subunit

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

High affinity binding of epibatidine to serotonin type 3 receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The role of palmitoylation in functional expression of nicotinic alpha7 receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Cys-loop neuroreceptors: structure to the rescue?

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Structure of the MscL homolog from Mycobacterium tuberculosis: a gated mechanosensitive ion channel

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

5-HT3 receptors are membrane ion channels

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

The role of loop 5 in acetylcholine receptor channel gating.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Crystal structure of acetylcholine-binding protein from Bulinus truncatus reveals the conserved structural scaffold and sites of variation in nicotinic acetylcholine receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Crystal structure of nicotinic acetylcholine receptor homolog AChBP in complex with an alpha-conotoxin PnIA variant.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Nicotine and carbamylcholine binding to nicotinic acetylcholine receptors as studied in AChBP crystal structures

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Gating mechanisms in Cys-loop receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A novel hyperekplexia-causing mutation in the pre-transmembrane segment 1 of the human glycine receptor alpha1 subunit reduces membrane expression and impairs gating by agonists.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Using physical chemistry to differentiate nicotinic from cholinergic agonists at the nicotinic acetylcholine receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Characterization of the effects of charged residues in the intracellular loop on ion permeation in alpha1 glycine receptor channels.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Charged residues at the 2' position of human GABAC rho 1 receptors invert ion selectivity and influence open state probability

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A single residue in the M2-M3 loop is a major determinant of coupling between binding and gating in neuronal nicotinic receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A point mutation in the gamma2 subunit of gamma-aminobutyric acid type A receptors results in altered benzodiazepine binding site specificity

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Subtle changes in residue 77 of the gamma subunit of alpha1beta2gamma2 GABAA receptors drastically alter the affinity for ligands of the benzodiazepine binding site

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Importance of the C-terminus of the human 5-HT3A receptor subunit

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

A Hydrophobic Gating Mechanism for Nanopores

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Acetylcholine receptor channel imaged in the open state

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

Patch-clamp fluorometry recording of conformational rearrangements of ion channels

21 January 2018

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Spatial orientation of the antagonist granisetron in the ligand-binding site of the 5-HT3 receptor

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Nicotinic acetylcholine receptor at 9 A resolution.

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Subunit counting in membrane-bound proteins

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

A (beta)-strand in the (gamma)2 subunit lines the benzodiazepine binding site of the GABA A receptor: structural rearrangements detected during channel gating.

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Mechanism of Cl- selection by a glutamate-gated chloride (GluCl) receptor revealed through mutations in the selectivity filter

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Dynamic modification of a mutant cytoplasmic cysteine residue modulates the conductance of the human 5-HT3A receptor

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Structural determinants of fast desensitization and desensitization-deactivation coupling in GABAa receptors.

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Subunit composition of functional nicotinic receptors in dopaminergic neurons investigated with knock-out mice

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Two tyrosine residues on the alpha subunit are crucial for benzodiazepine binding and allosteric modulation of gamma-aminobutyric acidA receptors

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Effects of quinine, quinidine, and chloroquine on alpha9alpha10 nicotinic cholinergic receptors

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Evidence for a centrally located gate in the pore of a serotonin-gated ion channel.

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Transducing agonist binding to channel gating involves different interactions in 5-HT3 and GABAC receptors

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

On the nature of partial agonism in the nicotinic receptor superfamily

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Selective electrical silencing of mammalian neurons in vitro by the use of invertebrate ligand-gated chloride channels.

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

A single amino-acid in the TM1 domain is an important determinant of the desensitization kinetics of recombinant human and guinea pig alpha-homomeric 5-hydroxytryptamine type 3 receptors

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Identifying the lipid-protein interface of the Torpedo nicotinic acetylcholine receptor: secondary structure implications

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Fluorescence techniques for fundamental and applied studies of membrane protein receptors: the 5-HT3 serotonin receptor

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Substitutions of the highly conserved M2 leucine create spontaneously opening rho1 gamma-aminobutyric acid receptors.

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Indazoles as indole bioisosteres: synthesis and evaluation of the tropanyl ester and amide of indazole-3-carboxylate as antagonists at the serotonin 5HT3 receptor

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Probing the structure of the nicotinic acetylcholine receptor with the hydrophobic photoreactive probes [125I]TID-BE and [125I]TIDPC/16

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Quantification of cation-pi interactions in protein-ligand complexes: crystal-structure analysis of Factor Xa bound to a quaternary ammonium ion ligand

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Identification of a Drosophila melanogaster glutamate-gated chloride channel sensitive to the antiparasitic agent avermectin

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Modified 5-HT3A receptor function by co-expression of alternatively spliced human 5-HT3A receptor isoforms

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

The surface accessibility of the glycine receptor M2-M3 loop is increased in the channel open state.

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Pore size and negative charge as structural determinants of permeability in the Torpedo nicotinic acetylcholine receptor channel

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Photoaffinity labeling of the benzodiazepine binding site of alpha1beta3gamma2 gamma-aminobutyric acidA receptors with flunitrazepam identifies a subset of ligands that interact directly with His102 of the alpha subunit and predicts orientation of t

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Anion permeation in GABA- and glycine-gated channels of mammalian cultured hippocampal neurons

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Residues at positions 206 and 209 of the alpha1 subunit of gamma-aminobutyric AcidA receptors influence affinities for benzodiazepine binding site ligands

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

The role of an alpha subtype M2-M3 His in regulating inhibition of GABAA receptor current by zinc and other divalent cations

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Rapid seizure-induced reduction of benzodiazepine and Zn2+ sensitivity of hippocampal dentate granule cell GABAA receptors

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Protein mobility and GABA-induced conformational changes in GABA(A) receptor pore-lining M2 segment

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Determinants of zinc potentiation on the alpha4 subunit of neuronal nicotinic receptors

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Conserved phosphorylation of the intracellular domains of GABA(A) receptor beta2 and beta3 subunits by cAMP-dependent protein kinase, cGMP-dependent protein kinase protein kinase C and Ca2+/calmodulin type II-dependent protein kinase

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Functional properties of a cloned 5-hydroxytryptamine ionotropic receptor subunit: comparison with native mouse receptors

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Rings of anionic amino acids as structural determinants of ion selectivity in the acetylcholine receptor channel

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Structure and dynamics of the pore-lining helix of the nicotinic receptor: MD simulations in water, lipid bilayers, and transbilayer bundles

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Mutational analysis of the charge selectivity filter of the alpha7 nicotinic acetylcholine receptor

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Phosphorylation of the predicted major intracellular domains of the rat and chick neuronal nicotinic acetylcholine receptor alpha 7 subunit by cAMP-dependent protein kinase

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

Secondary structure analysis of individual transmembrane segments of the nicotinic acetylcholine receptor by circular dichroism and Fourier transform infrared spectroscopy

1 reference

https://api.crossref.org/works/10.1017%2FS0033583510000168

7 January 2021

10.1017/S0033583510000168

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20849671%20AND%20SRC:MED&resulttype=core&format=json

release_tn4vtpoqcjajlhll7r7sibf5n4

14 February 2020

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/tn4vtpoqcjajlhll7r7sibf5n4

24 November 2022

mapped directly with Wikidata item

1 reference