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English
New paradigms in GPCR drug discovery.
scientific article published on 08 August 2015
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scholarly article
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Europe PubMed Central
PMC publication ID
4967540
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26265138%20AND%20SRC:MED&resulttype=core&format=json
retrieved
22 February 2020
review article
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stated in
Europe PubMed Central
title
New paradigms in GPCR drug discovery
(English)
1 reference
stated in
Europe PubMed Central
PMC publication ID
4967540
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26265138%20AND%20SRC:MED&resulttype=core&format=json
retrieved
22 February 2020
main subject
G protein-coupled receptor
0 references
drug discovery
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based on heuristic
inferred from title
author
Kenneth A. Jacobson
series ordinal
1
1 reference
stated in
Europe PubMed Central
PMC publication ID
4967540
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26265138%20AND%20SRC:MED&resulttype=core&format=json
retrieved
22 February 2020
author name string
Kenneth A Jacobson
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1
1 reference
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Europe PubMed Central
PMC publication ID
4967540
retrieved
18 August 2017
language of work or name
English
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publication date
8 August 2015
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Europe PubMed Central
PMC publication ID
4967540
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26265138%20AND%20SRC:MED&resulttype=core&format=json
retrieved
22 February 2020
published in
Biochemical Pharmacology
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stated in
Europe PubMed Central
PMC publication ID
4967540
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26265138%20AND%20SRC:MED&resulttype=core&format=json
retrieved
22 February 2020
volume
98
1 reference
stated in
Europe PubMed Central
PMC publication ID
4967540
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26265138%20AND%20SRC:MED&resulttype=core&format=json
retrieved
22 February 2020
issue
4
1 reference
stated in
Europe PubMed Central
PMC publication ID
4967540
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26265138%20AND%20SRC:MED&resulttype=core&format=json
retrieved
22 February 2020
page(s)
541-555
1 reference
stated in
Europe PubMed Central
PMC publication ID
4967540
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26265138%20AND%20SRC:MED&resulttype=core&format=json
retrieved
22 February 2020
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6 September 2017
Label-free drug discovery
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GPCR-targeting nanobodies: attractive research tools, diagnostics, and therapeutics
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GPCR signaling along the endocytic pathway
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Tuning up the right signal: chemical and genetic approaches to study GPCR functions
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6 September 2017
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6 September 2017
Targeting a G-protein-coupled receptor overexpressed in endocrine tumors by magnetic nanoparticles to induce cell death
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Combining on-chip synthesis of a focused combinatorial library with computational target prediction reveals imidazopyridine GPCR ligands
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6 September 2017
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The β-arrestin-biased ligand TRV120023 inhibits angiotensin II-induced cardiac hypertrophy while preserving enhanced myofilament response to calcium
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6 September 2017
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6 September 2017
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6 September 2017
Structural Features for Functional Selectivity at Serotonin Receptors
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Biophysical Fragment Screening of the β 1 -Adrenergic Receptor: Identification of High Affinity Arylpiperazine Leads Using Structure-Based Drug Design
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6 September 2017
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6 September 2017
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6 September 2017
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In vitro and in vivo antagonism of a G protein-coupled receptor (S1P3) with a novel blocking monoclonal antibody
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6 September 2017
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6 September 2017
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Small molecule disruption of G beta gamma signaling inhibits the progression of heart failure
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Discovery of the dual orexin receptor antagonist [(7R)-4-(5-chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl]methanone (MK-4305) for the treatment of insomnia
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Brain adenosine A2A receptor occupancy by a novel A1/A2A receptor antagonist, ASP5854, in rhesus monkeys: relationship to anticataleptic effect
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Discovery of a novel, orally active himbacine-based thrombin receptor antagonist (SCH 530348) with potent antiplatelet activity
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Translocation of arrestin induced by human A(3) adenosine receptor ligands in an engineered cell line: comparison with G protein-dependent pathways
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Clinical evidence for utilization of the A3 adenosine receptor as a target to treat rheumatoid arthritis: data from a phase II clinical trial
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reference URL
https://pubmed.ncbi.nlm.nih.gov/26265138
retrieved
12 December 2020
based on heuristic
inferred from PubMed ID database lookup
Organic chemistry in drug discovery
1 reference
stated in
PubMed
reference URL
https://pubmed.ncbi.nlm.nih.gov/26265138
retrieved
12 December 2020
based on heuristic
inferred from PubMed ID database lookup
Genotype-based treatment of type 2 diabetes with an α2A-adrenergic receptor antagonist
1 reference
stated in
PubMed
reference URL
https://pubmed.ncbi.nlm.nih.gov/26265138
retrieved
12 December 2020
based on heuristic
inferred from PubMed ID database lookup
CrossTalk opposing view: Weighing the evidence for class A GPCR dimers, the jury is still out
1 reference
stated in
PubMed
reference URL
https://pubmed.ncbi.nlm.nih.gov/26265138
retrieved
12 December 2020
based on heuristic
inferred from PubMed ID database lookup
Identifiers
DOI
10.1016/J.BCP.2015.08.085
1 reference
stated in
Europe PubMed Central
PMC publication ID
4967540
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26265138%20AND%20SRC:MED&resulttype=core&format=json
retrieved
22 February 2020
PMC publication ID
4967540
1 reference
stated in
Europe PubMed Central
PMC publication ID
4967540
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26265138%20AND%20SRC:MED&resulttype=core&format=json
retrieved
22 February 2020
PubMed publication ID
26265138
1 reference
stated in
Europe PubMed Central
PMC publication ID
4967540
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26265138%20AND%20SRC:MED&resulttype=core&format=json
retrieved
22 February 2020
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