(Q36885247)

16 August 2017

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title

Prediction of human pharmacokinetics--gastrointestinal absorption (English)

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16 August 2017

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Urban Fagerholm

1

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16 August 2017

publication date

1 July 2007

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Journal of Pharmacy and Pharmacology

16 August 2017

published in

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16 August 2017

volume

59

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16 August 2017

issue

7

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16 August 2017

page(s)

905-916

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Predicting the impact of physiological and biochemical processes on oral drug bioavailability

16 August 2017

cites work

1 reference

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Caco-2 monolayers in experimental and theoretical predictions of drug transport

21 January 2018

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Cell culture-based models for intestinal permeability: a critique

21 January 2018

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In silico predictions of drug solubility and permeability: two rate-limiting barriers to oral drug absorption

21 January 2018

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Why is it challenging to predict intestinal drug absorption and oral bioavailability in human using rat model.

21 January 2018

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Linear correlation of the fraction of oral dose absorbed of 64 drugs between humans and rats

21 January 2018

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https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Evaluation of using dog as an animal model to study the fraction of oral dose absorbed of 43 drugs in humans.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Comparison of oral absorption and bioavailablity of drugs between monkey and human

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Rapid calculation of polar molecular surface area and its application to the prediction of transport phenomena. 1. Prediction of intestinal absorption

21 January 2018

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Predicting passive transport in silico--history, hype, hope

21 January 2018

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Development and evaluation of an in vitro method for prediction of human drug absorption II. Demonstration of the method suitability.

21 January 2018

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Absorption potential: estimating the fraction absorbed for orally administered compounds

21 January 2018

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Dissolution testing as a prognostic tool for oral drug absorption: immediate release dosage forms

21 January 2018

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Evaluation and suggested improvements of the Biopharmaceutics Classification System (BCS).

21 January 2018

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Clinical pharmacokinetics of the cyclooxygenase inhibiting nitric oxide donator (CINOD) AZD3582.

21 January 2018

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Comparison between permeability coefficients in rat and human jejunum

21 January 2018

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Jejunal permeability in humans in vivo and rats in situ: investigation of molecular size selectivity and solvent drag

21 January 2018

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Pre-clinical pharmacokinetics of the cyclooxygenase-inhibiting nitric oxide donor (CINOD) AZD3582.

21 January 2018

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Drug permeability across a phospholipid vesicle based barrier: a novel approach for studying passive diffusion.

21 January 2018

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Physiologically-based pharmacokinetic simulation modelling.

21 January 2018

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Influence of physicochemical properties on dissolution of drugs in the gastrointestinal tract

21 January 2018

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MDCK (Madin-Darby canine kidney) cells: A tool for membrane permeability screening

21 January 2018

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Prediction of human drug clearance from in vitro and preclinical data using physiologically based and empirical approaches

21 January 2018

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Quantitative prediction of in vivo drug clearance and drug interactions from in vitro data on metabolism, together with binding and transport

21 January 2018

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Prediction of in vivo drug metabolism in the human liver from in vitro metabolism data

21 January 2018

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Guidance in the setting of drug particle size specifications to minimize variability in absorption

21 January 2018

1 reference

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Comparison of the gastrointestinal anatomy, physiology, and biochemistry of humans and commonly used laboratory animals

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Molecular properties of WHO essential drugs and provisional biopharmaceutical classification

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

In vitro system to evaluate oral absorption of poorly water-soluble drugs: simultaneous analysis on dissolution and permeation of drugs

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Forecasting the oral absorption behavior of poorly soluble weak bases using solubility and dissolution studies in biorelevant media

21 January 2018

1 reference

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The use of biopharmaceutic classification of drugs in drug discovery and development: current status and future extension

21 January 2018

1 reference

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Characterization of fluids from the stomach and proximal jejunum in men and women.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Drug-like properties and the causes of poor solubility and poor permeability

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Exploring the role of different drug transport routes in permeability screening.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

pH-dependent bidirectional transport of weakly basic drugs across Caco-2 monolayers: implications for drug-drug interactions.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Polar molecular surface properties predict the intestinal absorption of drugs in humans.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Prediction of intestinal absorption: comparative assessment of GASTROPLUS and IDEA.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Quantitative biopharmaceutics classification system: the central role of dose/solubility ratio.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Evaluation of a single-pass intestinal-perfusion method in rat for the prediction of absorption in man.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Variability in mRNA expression of ABC- and SLC-transporters in human intestinal cells: comparison between human segments and Caco-2 cells.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Prediction of hepatic clearance and availability by cryopreserved human hepatocytes: an application of serum incubation method

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Oral absorption of poorly water-soluble drugs: computer simulation of fraction absorbed in humans from a miniscale dissolution test.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Prediction of the oral absorption of low-permeability drugs using small intestine-like 2/4/A1 cell monolayers

21 January 2018

1 reference

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An improved cell culture model based on 2/4/A1 cell monolayers for studies of intestinal drug transport: characterization of transport routes.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Enzyme-catalyzed processes of first-pass hepatic and intestinal drug extraction

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Membrane transport of drugs in different regions of the intestinal tract of the rat.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

A comprehensive quantitative and qualitative evaluation of extrapolation of intravenous pharmacokinetic parameters from rat, dog, and monkey to humans. I. Clearance.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

A physiological model for the estimation of the fraction dose absorbed in humans.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Predicting drug disposition via application of BCS: transport/absorption/ elimination interplay and development of a biopharmaceutics drug disposition classification system

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

A 'rule of unity' for human intestinal absorption

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Correlating partitioning and caco-2 cell permeability of structurally diverse small molecular weight compounds

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

The "high solubility" definition of the current FDA Guidance on Biopharmaceutical Classification System may be too strict for acidic drugs

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Transport approaches to the biopharmaceutical design of oral drug delivery systems: prediction of intestinal absorption

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Evaluation of human intestinal absorption data and subsequent derivation of a quantitative structure-activity relationship (QSAR) with the Abraham descriptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

Evaluation of rat intestinal absorption data and correlation with human intestinal absorption

21 January 2018

1 reference

https://api.crossref.org/works/10.1211%2FJPP.59.7.0001

21 January 2018

Identifiers

DOI

10.1211/JPP.59.7.0001

1 reference

release_4ob7lztgozhcvi7xxbx4nr357e

16 August 2017

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/4ob7lztgozhcvi7xxbx4nr357e

mapped directly with Wikidata item

24 November 2022

based on heuristic

1 reference